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PENTAZOCINE
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DeCS
Descriptor
English
:
Pentazocine
Descriptor
Spanish
:
Pentazocina
Descriptor
Portuguese
:
Pentazocina
Tree Number:
D03.132.577.249.106.700
D04.615.723.795.106.700
Definition
English
:
The first mixed agonist-antagonist analgesic to be marketed. It is an agonist at the kappa and sigma opioid receptors and has a weak antagonist action at the mu receptor. (From AMA Drug Evaluations Annual, 1991, p97)
Pharmacological Action:
Adjuvants, Anesthesia
Analgesics, Opioid
Narcotic Antagonists
Narcotics
History Note
English
:
66(64)
Allowable Qualifiers
English
:
analogs & derivatives
administration & dosage
adverse effects
agonists
antagonists & inhibitors
analysis
blood
cerebrospinal fluid
chemistry
classification
chemical synthesis
contraindications
diagnostic use
economics
history
immunology
isolation & purification
metabolism
pharmacology
pharmacokinetics
poisoning
radiation effects
supply & distribution
standards
toxicity
therapeutic use
urine
Record Number:
10617
Unique Identifier:
D010423
Occurrence in VHL
:
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