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THIORPHAN
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DeCS
Descriptor
English
:
Thiorphan
Descriptor
Spanish
:
Tiorfan
Descriptor
Portuguese
:
Tiorfano
Tree Number:
D02.886.030.893
D12.125.166.893
D12.125.481.700.750
Definition
English
:
A potent inhibitor of membrane metalloendopeptidase (ENKEPHALINASE).
Thiorphan
potentiates morphine-induced
ANALGESIA
and attenuates naloxone-precipitated withdrawal
symptoms.
Pharmacological Action:
Protease Inhibitors
History Note
English
:
89
Allowable Qualifiers
English
:
analogs & derivatives
administration & dosage
adverse effects
agonists
antagonists & inhibitors
analysis
blood
cerebrospinal fluid
chemistry
classification
chemical synthesis
contraindications
diagnostic use
economics
history
immunology
isolation & purification
metabolism
pharmacology
pharmacokinetics
poisoning
radiation effects
supply & distribution
standards
toxicity
therapeutic use
urine
Record Number:
23847
Unique Identifier:
D015244
Occurrence in VHL
:
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